name: US9676701, 9 (trans)-2-(6-(4-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 10 (trans)-2-(6-(4-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 11 (trans)-2-(6-(3-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 12 4-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)benzonitrile dihydrochloride


name: US9676701, 13 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)benzonitrile hydrochloride


name: US9676701, 14 (Trans)-2-(6-p-tolylpyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 15 (Trans)-2-(6-m-tolylpyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 17 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenol dihydrochloride


name: US9676701, 19 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)benzamide hydrochloride


name: US9676701, 22 (trans)-2-(6-(3-methoxy-4-methylphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 23 5-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-2-fluorophenol hydrochloride


name: US9676701, 24 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-5-fluorophenol hydrochloride


name: US9676701, 25 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-4-fluorophenol hydrochloride


name: US9676701, 26 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-2-fluorophenol hydrochloride


name: US9676701, 29 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-5-chlorophenol hydrochloride


name: US9676701, 30 (trans)-2-(6-(2-fluoro-3-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 31 (trans)-2-(6-(5-chlorothiophen-2-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 34 (trans)-2-(6-(benzo[b]thiophen-5-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 38 (trans)-2-(6-(4-fluoro-3-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 39 (trans)-2-(6-(3-fluoro-5-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 40 (trans)-2-(6-(2-fluoro-5-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 41 (trans)-2-(6-(2-fluoro-3-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 42 (trans)-2-(6-(3-chloro-5-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 43 (trans)-2-(6-(2-chloro-5-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 44 (trans)-2-(6-(3-methoxy-5-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 45 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-5-methoxybenzonitrile hydrochloride


name: US9676701, 46 5-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-2-methylphenol hydrochloride


name: US9676701, 47 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-4-chlorophenol hydrochloride


name: US9676701, 48 3-(5-((trans)-2-amninocyclopropyl)pyridin-2-yl)-5-(trifluoromethyl)phenol hydrochloride


name: US9676701, 49 (trans)-2-(6-(2-fluoro-5-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 50 (trans)-2-(6-(2-chloro-5-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 51 (trans)-2-(6-(3,5-bis(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 52 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)acetamide hydrochloride


name: US9676701, 53 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)methanesulfonamide hydrochloride


name: US9676701, 54 (trans)-2-(6-(benzo[b]thiophen-2-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 55 (trans)-2-(6-(benzo[b]thiophen-3-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 56 5-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)thiophene-2-carbonitrile hydrochloride


name: US9676701, 57 (trans)-2-(6-(4-methylthiophen-3-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 58 (Trans)-2-(6-(3,4-difluoro-5-methoxyphenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 59 5-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-2,3-difluorophenol hydrochloride


name: US9676701, 60 (Trans)-2-(6-(1H-indazol-6-yl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 62 6-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)indolin-2-one hydrochloride


name: US9676701, 64 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)benzenesulfonamide hydrochloride


name: US9676701, 65 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)propane-2-sulfonamide hydrochloride


name: US9676701, 66 4'-((trans)-2-aminocyclopropyl)-4-fluorobiphenyl-3-ol hydrochloride


name: US9676701, 67 4'-((trans)-2-aminocyclopropyl)-5-chlorobiphenyl-3-ol hydrochloride


name: US9676701, 68 N-(4'-((trans)-2-aminocyclopropyl)biphenyl-3-yl)benzenesulfonamide hydrochloride


name: US9676701, 70 N-(4'-((trans)-2-aminocyclopropyl)biphenyl-3-yl)methanesulfonamide hydrochloride


name: US9676701, 71 N-(2-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)methanesulfonamide hydrochloride


name: US9676701, 72 3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-4-methoxybenzonitrile hydrochloride


name: US9676701, 73 N-(4'-((trans)-2-aminocyclopropyl)biphenyl-2-yl)methanesulfonamide hydrochloride


name: US9676701, 74 4'-((trans)-2-aminocyclopropyl)-6-methoxybiphenyl-3-carbonitrile hydrochloride


name: US9676701, 75 N-(4'-((trans)-2-aminocyclopropyl)-6-methoxybiphenyl-3-yl)methanesulfonamide hydrochloride


name: US9676701, 76 (trans)-2-(2-chloro-6-(3-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 80 (trans)-2-(2-methyl-6-(3-(trifluoromethyl)phenyl)pyridin-3-yl)cyclopropanamine hydrochloride


name: US9676701, 87 4'-((trans)-2-aminocyclopropyl)-6-hydroxybiphenyl-3-carbonitrile hydrochloride


name: US9676701, 88 N-(4'-((trans)-2-aminocyclopropyl)-6-hydroxybiphenyl-3-yl)methanesulfonamide hydrochloride


name: US9676701, 93 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-4-methoxyphenyl)methanesulfonamide hydrochloride


name: US9676701, 94 N-(4'-((trans)-2-aminocyclopropyl)-5-chloro-[1,1'-biphenyl]-3-yl)methanesulfonamide hydrochloride


name: US9676701, 95 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-5-chlorophenyl)methanesulfonamide hydrochloride


name: US9676701, 96 N-(4'-((trans)-2-aminocyclopropyl)-4-fluoro-[1,1'-biphenyl]-3-yl)methanesulfonamide hydrochloride


name: US9676701, 97 N-(5-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)-2-fluorophenyl)methanesulfonamide hydrochloride


name: US9676701, 98 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)ethanesulfonamide hydrochloride


name: US9676701, 99 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)-4-cyanobenzenesulfonamide hydrochloride


name: US9676701, 100 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)-3-cyanobenzenesulfonamide hydrochloride


name: US9676701, 101 N-(3-(5-((trans)-2-aminocyclopropyl)pyridin-2-yl)phenyl)-2-cyanobenzenesulfonamide hydrochloride


name: US9676701, 103 N-(4'-((trans)-2-aminocyclopropyl)-[1,1'-biphenyl]-3-yl)-1,1,1-trifluoromethanesulfonamide hydrochloride


name: US9676701, 104 4'â??((trans)-2-aminocyclopropyl)-6-hydroxy-[1,1'-biphenyl]-3-carbonitrile hydrochloride


name: US9676701, 105 4'-((trans)-2-aminocyclopropyl)-[1,1'-biphenyl]-2-ol hydrochloride


name: US9676701, 106 4'-((trans)-2-aminocyclopropyl)-3'-methoxy-[1,1'-biphenyl]-3-ol hydrochloride


name: US9676701, 113 3-(5-((trans)-2-aminocyclopropyl)thiophen-2-yl)phenol trihydrochloride


name: US9676701, 116 3-(5-((trans)-2-aminocyclopropyl)thiazol-2-yl)phenol hydrochloride


name: US9676701, 124 N-(3-(5-((trans)-2-aminocyclopropyl)thiazol-2-yl)phenyl)-2-cyanobenzenesulfonamide dihydrochloride


name: US9676728, 12-D (A) (+/-)-2-((2,6-Dimethoxy-4-methylphenyl)(methylamino)methyl)-1H-benzo[d]imidazole-5-carbonitrile


name: US9669031, 6 6'-(pyrimidin-4-ylamino)-1'H-spiro[cyclopentane-1,3'-imidazo[1,5-a]pyridine]-1',5'(2'H)-dione (Cpd. No. 6)


name: US9669031, 7 3-methyl-6-(pyrimidin-4-ylamino)-3-(2,2,2-trifluoroethyl)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 7)


name: US9669031, 8 3-isopropyl-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 8)


name: US9669031, 9 3-cyclopentyl-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 9)


name: US9669031, 10 N-(6-((3,3-dimethyl-1,5-dioxo-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 10)


name: US9669031, 11 3-(4-fluorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 11)


name: US9669031, 12 3-(3-fluorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 12)


name: US9669031, 13 3-(4-chlorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 13)


name: US9669031, 14 3-methyl-6-(pyrimidin-4-ylamino)-3-(trifluoromethyl)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 14)


name: US9669031, 16 3-methyl-6-(pyrimidin-4-ylamino)-3-(thiophen-3-yl)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 16)


name: US9669031, 18 3-(3-chlorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 18)


name: US9669031, 20 6-(pyrimidin-4-ylamino)-1H-spiro[imidazo[1,5-a]pyridine-3,3'-piperidine]-1,5(2H)-dione (Cpd. No. 20)


name: US9669031, 21 N-[6-[(1,5-dioxospiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclopentane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 21)


name: US9669031, 22 N-(6-((3-methyl-1,5-dioxo-3-(2,2,2-trifluoroethyl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 22)


name: US9669031, 23 N-[6-[(3-cyclopentyl-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 23)


name: US9669031, 24 N-[6-[[3-methyl-1,5-dioxo-3-(trifluoromethyl)-2H-imidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 24)


name: US9669031, 27 3-(3,5-difluorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 27)


name: US9669031, 28 3-(3-chloro-5-fluorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 28)


name: US9669031, 29 N-[6-[(3-isopropyl-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 29)


name: US9669031, 30 N-[6-[[3-(3-fluorophenyl)-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 30)


name: US9669031, 31 6-[[6-[(E)-2-cyclopropylvinyl]pyrimidin-4-yl]amino]-3-methyl-3-(trifluoromethyl)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 31)


name: US9669031, 33 3-(3,5-dichlorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 33)


name: US9669031, 34 3-methyl-3-(pyridin-2-yl)-6-(pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 34)


name: US9669031, 35 8-chloro-3-methyl-6-(pyrimidin-4-ylamino)-3-(trifluoromethyl)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 35)


name: US9669031, 36 2',2'-dimethyl-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclopentane]-1,5-dione (Cpd. No. 36)


name: US9669031, 37 6-[(8-cyclopropyl-9H-purin-6-yl)amino]-3-methyl-3-(trifluoromethyl)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 37)


name: US9669031, 38 N-[6-[(8-chloro-1,5-dioxo-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclopentane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 38)


name: US9669031, 39 8'-chloro-6'-(pyrimidin-4-ylamino)-2'H-spiro[cyclopentane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 39)


name: US9669031, 41 3-(2-aminoethyl)-3-methyl-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 41)


name: US9669031, 42 N-[6-[(8-chloro-3-cyclopentyl-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 42)


name: US9669031, 43 N-[6-[(8-chloro-3,3-dimethyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 43)


name: US9669031, 44 N-(6-((8'-chloro-1',5'-dioxo-1',5'-dihydro-2'H-spiro[cyclobutane-1,3'-imidazo[1,5-a]pyridin]-6'-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 44)


name: US9669031, 207 6'-((6-aminopyrimidin-4-yl)amino)-8'-(hydroxymethyl)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 207)


name: US9669031, 46 N-[6-[[8-chloro-3-methyl-1,5-dioxo-3-(2,2,2-trifluoroethyl)-2H-imidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 46)


name: US9669031, 48 8-chloro-3-cyclopentyl-3-methyl-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 48)


name: US9669031, 49 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-(trifluoromethyl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 49)


name: US9669031, 50 N-[6-[(8-chloro-4',4'-difluoro-1,5-dioxo-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 50)


name: US9669031, 51 N-[6-[[8-chloro-3-(3-chlorophenyl)-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 51)


name: US9669031, 53 (3'S)-3'-amino-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 53)


name: US9669031, 55 8-chloro-3-methyl-6-(pyrimidin-4-ylamino)-3-(2,2,2-trifluoroethyl)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 55)


name: US9669031, 56 N-(6-((8-chloro-1,5-dioxo-1,5-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidin]-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide hydrochloride (Cpd. No. 56)


name: US9669031, 57 8-chloro-3-(3-fluorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 57)


name: US9669031, 58 8-chloro-3-(3-chlorophenyl)-3-methyl-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 58)


name: US9669031, 59 6-((6-((1-cyclopropyl-2,2,2-trifluoroethyl)amino)pyrimidin-4-yl)amino)-3-methyl-3-(trifluoromethyl)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 59)


name: US9669031, 60 N-(6-((8-chloro-1,5-dioxo-1,5-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,3'-piperidin]-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide hydrochloride (Cpd. No. 60)


name: US9669031, 61 N-(6-((8-chloro-1,5-dioxo-1,2',3',5,5',6'-hexahydro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-pyran]-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 61)


name: US9669031, 62 N-[6-[(8-chloro-1',1'-difluoro-1,5-dioxo-spiro[2H-imidazo[1,5-a]pyridine-3,3'-cyclobutane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 62)


name: US9669031, 63 8-chloro-2',2'-dimethyl-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1, 5-a]pyridine-3,1'-cyclopentane]-1,5-dione (Cpd. No. 63)


name: US9669031, 64 8-chloro-6-(pyrimidin-4-ylamino)-2',3',5',6'-tetrahydro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-pyran]-1,5-dione (Cpd. No. 64)


name: US9669031, 65 N-(6-((8-chloro-1,5-dioxo-1,5-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,3'-thietan]-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 65)


name: US9669031, 66 8-chloro-2'-fluoro-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 66)


name: US9669031, 69 8-fluoro-3,3-dimethyl-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 69)


name: US9669031, 70 6'-((6-aminopyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 70)


name: US9669031, 72 8-chloro-3-methyl-3-(3-pyridyl)-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 72)


name: US9669031, 73 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-(pyridin-4-yl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 73)


name: US9669031, 74 8-chloro-3-methyl-3-(2-pyridyl)-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 74)


name: US9669031, 75 8-chloro-3-methyl-3-(4-pyridyl)-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 75)


name: US9669031, 76 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-(pyridin-2-yl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 76)


name: US9669031, 77 N-[6-[[8-chloro-3-methyl-1,5-dioxo-3-(3-pyridyl)-2H-imidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 77)


name: US9669031, 78 N-(6-((8'-chloro-2-fluoro-1',5'-dioxo-1',5'-dihydro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridin]-6'-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 78)


name: US9669031, 80 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-(3-(trifluoromethyl)phenyl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 80)


name: US9669031, 83 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-(m-tolyl)-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 83)


name: US9669031, 84 N-[6-[(3-tert-butyl-8-chloro-3-methyl-1,5-dioxo-2H-imidazo[1,5-a]pyridin-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 84)


name: US9669031, 85 N-[6-[[8-chloro-1,5-dioxo-3-(trifluoromethyl)-2,3-dihydroimidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 85)


name: US9669031, 86 N-[6-[(8-chloro-1,5-dioxo-spiro[2H-imidazo[1,5-a]pyridine-3,3'-azetidine]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide hydrochloride (Cpd. No. 86)


name: US9669031, 89 8-chloro-3-(3-chlorophenyl)-3-methyl-6-[[6-(methylamino)pyrimidin-4-yl]amino]-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 89)


name: US9669031, 90 8-chloro-3-methyl-3-(6-methyl-2-pyridyl)-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 90)


name: US9669031, 91 N-[6-[[8-chloro-3-(3-fluorophenyl)-1,5-dioxo-2,3-dihydroimidazo[1,5-a]pyridin-6-yl]amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 91)


name: US9669031, 92 6-[(6-aminopyrimidin-4-yl)amino]-3-(3-chlorophenyl)-3,8-dimethyl-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 92)


name: US9669031, 94 6-[(6-aminopyrimidin-4-yl)amino]-8-chloro-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclopentane]-1,5-dione (Cpd. No. 94)


name: US9669031, 95 N-[6-[(8-chloro-1,1',5-trioxo-spiro[2H-imidazo[1,5-a]pyridine-3,3'-thietane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide (Cpd. No. 95)


name: US9669031, 96 8-chloro-1',1'-dimethyl-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,2'-cyclohexane]-1,5-dione (Cpd. No. 96)


name: US9669031, 97 N-(6-((8-chloro-3-methyl-1,5-dioxo-3-phenyl-1,2,3,5-tetrahydroimidazo[1,5-a]pyridin-6-yl)amino)pyrimidin-4-yl)cyclopropanecarboxamide (Cpd. No. 97)


name: US9669031, 98 6-[(6-aminopyrimidin-4-yl)amino]-8-methyl-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclopentane]-1,5-dione hydrochloride (Cpd. No. 98)


name: US9669031, 100 8-chloro-6-((7-cyclopropylpyrido[4,3-d]pyrimidin-4-yl)amino)-3,3-dimethyl-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 100)


name: US9669031, 101 6-((6-aminopyrimidin-4-yl)amino)-3-(3-fluorophenyl)-3,8-dimethyl-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 101)


name: US9669031, 102 6-((6-aminopyrimidin-4-yl)amino)-3,3,8-trimethyl-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione hydrochloride (Cpd. No. 102)


name: US9669031, 103 6-[(6-aminopyrimidin-4-yl)amino]-4',4'-difluoro-8-methyl-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione hydrochloride (Cpd. No. 103)


name: US9669031, 104 8-chloro-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione hydrochloride (Cpd. No. 104)


name: US9669031, 105 6-[(6-aminopyrimidin-4-yl)amino]-3-tert-butyl-8-chloro-3-methyl-2H-imidazo[1,5-a]pyridine-1,5-dione hydrochloride (Cpd. No. 105)


name: US9669031, 106 6-((6-aminopyrimidin-4-yl)amino)-8-methyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione dihydrochloride (Cpd. No. 106)


name: US9669031, 107 6'-((6-aminopyrimidin-4-yl)amino)-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 107)


name: US9669031, 108 6-((6-aminopyrimidin-4-yl)amino)-8-chloro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione dihydrochloride (Cpd. No. 108)


name: US9669031, 109 8-chloro-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione hydrochloride (Cpd. No. 109)


name: US9669031, 110 8-chloro-4',4'-difluoro-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione hydrochloride (Cpd. No. 110)


name: US9669031, 111 6-[(6-aminopyrimidin-4-yl)amino]-6',8-dichloro-spiro[2H-imidazo[1,5-a]pyridine-3,1'-indane]-1,5-dione hydrochloride (Cpd. No. 111)


name: US9669031, 112 8-chloro-6-[(5-fluoropyrimidin-4-yl)amino]spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 112)


name: US9669031, 113 8-chloro-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,2'-indane]-1,1',5-trione (Cpd. No. 113)


name: US9669031, 114 6-((6-aminopyrimidin-4-yl)amino)-8-chloro-6'-fluoro-2',3'-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,1'-indene]-1,5-dione hydrochloride (Cpd. No. 114)


name: US9669031, 115 8-chloro-6-[(5-chloropyrimidin-4-yl)amino]spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 115)


name: US9669031, 116 8-chloro-6-[(6-methylpyrimidin-4-yl)amino]spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 116)


name: US9669031, 119 6-[(6-aminopyrimidin-4-yl)amino]-8-chloro-3-(3-fluorophenyl)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 119)


name: US9669031, 120 8'-chloro-2,2-dimethyl-6'-(pyrimidin-4-ylamino)-2'H-spiro[cyclobutane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 120)


name: US9669031, 121 6'-((6-Aminopyrimidin-4-yl)amino)-8'-chloro-2,2-dimethyl-2'H-spiro[cyclobutane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 121)


name: US9669031, 122 6-[(6-amino-5-chloro-pyrimidin-4-yl)amino]-8-chloro-spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione hydrochloride (Cpd. No. 122)


name: US9669031, 124 8-chloro-3,3-dimethyl-6-(pyrido[4,3-d]pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 124)


name: US9669031, 125 8'-chloro-6'-((2-methylpyrimidin-4-yl)amino)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 125)


name: US9669031, 126 6-((6-aminopyrimidin-4-yl)amino)-8-chloro-2H-spiro[imidazo[1,5-a]pyridine-3,6'-[1,4]diazepane]-1,5-dione (Cpd. No. 126)


name: US9669031, 128 6-[(6-aminopyrimidin-4-yl)amino]-8-chloro-1'-methyl-spiro[2H-imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione hydrochloride (Cpd. No. 128)


name: US9669031, 129 8-chloro-1'-methyl-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 129)


name: US9669031, 130 1',8-dimethyl-6-(pyrimidin-4-ylamino)-2H-spiro[imidazo[1,5-a]pyridine-3,3'-piperidine]-1,5-dione (Cpd. No. 130)


name: US9669031, 133 8'-chloro-6'-(pyrimidin-4-ylamino)-5'-thioxo-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridin]-1'(5'H)-one (Cpd. No. 133)


name: US9669031, 142 4-((8'-chloro-1',5'-dioxo-1',5'-dihydro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridin]-6'-yl)amino)pyrimidine-5-carbonitrile (Cpd. No. 142)


name: US9669031, 143 8'-chloro-6'-((5-(1-methyl-1H-pyrazol-4-yl)pyrimidin-4-yl)amino)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 143)


name: US9669031, 155 8-chloro-1'-(2-hydroxyethyl)-6-(pyrimidin-4-ylamino)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 155)


name: US9669031, 156 8-chloro-1'-(2,2-difluoroethyl)-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 156)


name: US9669031, 157 8-chloro-6-(pyrimidin-4-ylamino)-1'-(2,2,2-trifluoroethyl)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 157)


name: US9669031, 158 8'-chloro-8-methyl-6'-(pyrimidin-4-ylamino)-2'H-8-azaspiro[bicyclo[3.2.1]octane-3,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 158)


name: US9669031, 160 2-(8-chloro-1,5-dioxo-6-(pyrimidin-4-ylamino)-1,5-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidin]-1'-yl)acetonitrile (Cpd. No. 160)


name: US9669031, 162 8-chloro-4'-(methylamino)-6-(pyrimidin-4-ylamino)spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione hydrochloride (Cpd. No. 162)


name: US9669031, 163 1'-acetyl-8-chloro-6-(pyrimidin-4-ylamino)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 163)


name: US9669031, 164 8'-chloro-1',5'-dioxo-6'-(pyrimidin-4-ylamino)-1',5'-dihydro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-4-carbonitrile (Cpd. No. 164)


name: US9669031, 165 8-chloro-3,3-dimethyl-6-(pyrido[3,4-d]pyrimidin-4-ylamino)-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 165)


name: US9669031, 169 6'-((6-amino-5-fluoropyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 169)


name: US9669031, 170 6-[(6-aminopyrimidin-4-yl)amino]-1',8-dimethyl-spiro[2H-imidazo[1,5-a]pyridine-3,3'-piperidine]-1,5-dione (Cpd. No. 170)


name: US9669031, 187 8-chloro-6-[(5-methoxypyrimidin-4-yl)amino]spiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-1,5-dione (Cpd. No. 187)


name: US9669031, 188 6'-((6-amino-5-ethylpyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 188)


name: US9669031, 189 6'-((6-amino-5-isopropylpyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 189)


name: US9669031, 191 8'-chloro-6'-(pyrimidin-4-ylamino)-2-(trifluoromethyl)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 191)


name: US9669031, 192 8-chloro-3-methyl-3-(2-methylprop-1-enyl)-6-(pyrimidin-4-ylamino)-2H-imidazo[1,5-a]pyridine-1,5-dione (Cpd. No. 192)


name: US9669031, 193 6'-((6-amino-5-methylpyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 193)


name: US9669031, 194 8'-chloro-6'-((5-ethylpyrimidin-4-yl)amino)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 194)


name: US9669031, 195 6'-((6-amino-5-methoxypyrimidin-4-yl)amino)-8'-chloro-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 195)


name: US9669031, 196 8'-chloro-6'-((5-ethoxypyrimidin-4-yl)amino)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 196)


name: US9669031, 197 8'-chloro-6'-((5-isopropoxypyrimidin-4-yl)amino)-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 197)


name: US9669031, 204 6'-((6-aminopyrimidin-4-yl)amino)-2-hydroxy-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 204)


name: US9669031, 208 6'-((5-cyclopropylpyrimidin-4-yl)amino)-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 208)


name: US9669031, 213 5-((6-aminopyrimidin-4-yl)amino)-3-chloro-1-isobutyl-6-oxo-1,6-dihydropyridine-2-carboxamide (Cpd. No. 213)


name: US9669031, 215 3'-(pyrimidin-4-ylamino)-4'H-spiro[cyclohexane-1,6'-imidazo[1,5-a]pyrimidine]-4',8'(7'H)-dione (Cpd. No. 215)


name: US9669031, 219 6-((6-aminopyrimidin-4-yl)amino)-1',8-dimethyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione hydrochloride (Cpd. No. 219)


name: US9669031, 220 6-((6-amino-5-methylpyrimidin-4-yl)amino)-1',8-dimethyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 220)


name: US9669031, 222 6'-((6-amino-5-methylpyrimidin-4-yl)amino)-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 222)


name: US9669031, 223 6'-((6-amino-5-chloropyrimidin-4-yl)amino)-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione hydrochloride (Cpd. No. 223)


name: US9669031, 225 2-(6-((6-aminopyrimidin-4-yl)amino)-8-methyl-1,5-dioxo-1,5-dihydro-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidin]-1'-yl)acetonitrile (Cpd. No. 225)


name: US9669031, 226 6-((6-aminopyrimidin-4-yl)amino)-1'-(2,2-difluoroethyl)-8-methyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 226)


name: US9669031, 230 1'-(2,2-difluoroethyl)-6-((5-methoxypyrimidin-4-yl)amino)-8-methyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 230)


name: US9669031, 231 6'-((6-amino-5-methoxypyrimidin-4-yl)amino)-8'-methyl-2'H-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione (Cpd. No. 231)


name: US9669031, 232 6-((6-aminopyrimidin-4-yl)amino)-8-methyl-1'-(2,2,2-trifluoroethyl)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 232)


name: US9669031, 233 6-((6-amino-5-methylpyrimidin-4-yl)amino)-1'-(2,2-difluoroethyl)-8-methyl-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 233)


name: US9669031, 234 6-((6-amino-5-methoxypyrimidin-4-yl)amino)-8-methyl-1'-(2,2,2-trifluoroethyl)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 234)


name: US9669031, 235 6-((5-methoxypyrimidin-4-yl)amino)-8-methyl-1'-(2,2,2-trifluoroethyl)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 235)


name: US9669031, 236 6-((6-amino-5-methylpyrimidin-4-yl)amino)-8-methyl-1'-(2,2,2-trifluoroethyl)-2H-spiro[imidazo[1,5-a]pyridine-3,4'-piperidine]-1,5-dione (Cpd. No. 236)


name: US9670142, A5 4'-chloro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A8 biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A12 4'-cyano-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A16 5-benzoxazol-2-yl-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A17 5-benzoxazol-2-yl-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A39 (S)-2-acetylamino-N-{(1S,3R)-3-[(4-benzoxazol-2-yl-benzoyl)-methyl-amino]-cyclopentyl}-succinamic acid methyl ester


name: US9670142, A40 (R)-tetrahydro-furan-2-carboxylic acid {(1S,3R)-3-[(4-benzoxazol-2-yl-benzoyl)-methyl-amino]-cyclopentyl}-amide


name: US9670142, A41 (S)-tetrahydro-furan-2-carboxylic acid {(1S,3R)-3-[(4-benzoxazol-2-yl-benzoyl)-methyl-amino]-cyclopentyl}-amide


name: US9670142, A51 4'-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-biphenyl-4-carboxylic acid


name: US9670142, A52 3-methyl-4'-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-biphenyl-4-carboxylic acid


name: US9670142, A53 4'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A54 2'-fluoro-4'-(4-methyl-cyclohexyl)-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A55 tert-butyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A56 3',4'-dimethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A57 biphenyl-4,4'-dicarboxylic acid 4'-amide 4-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide]


name: US9670142, A61 4'-cyano-3',5'-difluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A62 4'-trifluoromethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A63 3'-chloro-4'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A64 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A65 4'-methoxy-2'-methyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A66 3'-fluoro-4'-methyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A68 4'-pyrazol-1-yl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A69 3-fluoro-4'-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-biphenyl-4-carboxylic acid methyl ester


name: US9670142, A70 4'-cyclopropylmethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A71 4'-cyano-3'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A73 4'-methyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A77 cyano-2'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A78 biphenyl-4,4'-dicarboxylic acid 4'-methylamide 4-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide]


name: US9670142, A79 fluoro-4'-trifluoromethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A81 4'-(2H-pyrazol-3-yl)-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A82 4'-methoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A83 2',4'-difluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A85 4'-difluoromethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A86 4'-chloro-3'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A88 2',4'-dimethoxy-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A89 4'-(5-propyl-tetrahydro-pyran-2-yl)-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A90 2',4'-dimethyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A92 4'-chloro-2'-fluoro-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A96 4'-isopropyl-biphenyl-4-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A97 2-fluoro-4'-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-biphenyl-4-carboxylic acid methyl ester


name: US9670142, A103 5-(6-methyl-1H-indazol-5-yl)-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A104 5-(7-methyl-1H-indazol-5-yl)-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A105 5-(3-methyl-1H-indazol-5-yl)-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A109 5-(1H-indol-5-yl)-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A110 5-(1-methyl-1H-indol-5-yl)-pyridine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A113 6-(1H-indol-5-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A118 6-(1-methyl-1H-indol-5-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A125 5-(1-methyl-1H-indol-5-yl)-pyrazine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A131 5-(1H-indol-5-yl)-pyrimidine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A132 5-(1H-indol-5-yl)-pyrazine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A133 5-(1-methyl-1H-indol-5-yl)-pyrimidine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A136 6-(7-fluoro-1H-indol-5-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A137 6-(4-fluoro-1H-indol-5-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A138 (S)-tetrahydro-furan-2-carboxylic acid ((1S,3R)-3-{[4-(6-chloro-benzooxazol-2-yl)-benzoyl]-methyl-amino}-cyclopentyl)-amide


name: US9670142, A139 2-(1H-indol-5-yl)-pyrimidine-5-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A148 5-(6-chloro-benzoxazol-2-yl)-pyrazine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A149 5-(6-chloro-benzoxazol-2-yl)-pyrimidine-2-carboxylic acid methyl-{(1R,3S)-3-[((S)-tetrahydro-furan-2-carbonyl)-amino]-cyclopentyl}-amide


name: US9670142, A150 6-(4-methyl-1H-indol-5-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A155 6-(6-chloro-benzoxazol-2-yl)-pyridazine-3-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A156 5-(6-chloro-benzoxazol-2-yl)-pyrimidine-2-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A159 5-(6-chloro-benzoxazol-2-yl)-pyrazine-2-carboxylic acid methyl-{(1R,3S)-3-[((S)-tetrahydro-furan-2-carbonyl)-amino]-cyclopentyl}-amide


name: US9670142, A160 5-{2-fluoro-4-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-phenyl}-1H-indole-3-carboxylic acid amide


name: US9670142, A170 2-(1H-indol-5-yl)-thiazole-5-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A171 7-fluoro-5-{4-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-phenyl}-1H-indole-3-carboxylic acid amide


name: US9670142, A172 7-fluoro-5-{2-fluoro-4-[methyl-((1R,3S)-3-propionylamino-cyclopentyl)-carbamoyl]-phenyl}-1H-indole-3-carboxylic acid amide


name: US9670142, A173 2-(1H-indol-5-yl)-4-methyl-thiazole-5-carboxylic acid methyl-((1R,3S)-3-propionylamino-cyclopentyl)-amide


name: US9670142, A174 (S)-tetrahydro-furan-2-carboxylic acid ((1S,3R)-3-{-([4-(5-chloro-benzoxazol-2-yl)-benzoyl]-methyl-amino}-cyclopentyl)-amide


name: US9670142, A175 (S)-tetrahydro-furan-2-carboxylic acid {(1S,3R)-3-[(4-benzoxazol-2-yl-2-fluoro-benzoyl)-methyl-amino]-cyclopentyl}-amide


name: US9670157, 1 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 2 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 3 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 4 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 8 2,5-Dimethyl-1-(5-pyridin-3-yl-thiophen-3-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 9 2,5-Dimethyl-1-(4-phenyl-thiophen-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 10 2,5-Dimethyl-1-(5-phenyl-thiophen-3-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 11 2,5-Dimethyl-1-(3-phenyl-isoxazol-5-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 12 1-Benzothiazol-2-ylmethyl-2,5-dimethyl-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 14 2,5-Dimethyl-1-(4-pyridin-4-yl-thiophen-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 15 2,5-Dimethyl-1-(6-morpholin-4-yl-pyridin-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 16 2,5-Dimethyl-1-(6-phenyl-pyridin-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 17 1-[2,3']Bipyridinyl-6-ylmethyl-2,5-dimethyl-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 18 2,5-Methyl-1-(2-phenyl-oxazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 20 2,5-Dimethyl-1-thiophen-2-ylmethyl-1H-pyrrole-3-carboxylic acid4-amidomethyl-benzylamide


name: US9670157, 21 2,5-Dimethyl-1-(5-pyridin-4-yl-thiophen-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 22 2,5-Dimethyl-1-(5-phenyl-thiophen-2-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 23 2,5-Dimethyl-1-[5-(2-methyl-thiazol-4-yl)-thiophen-2-ylmethyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 24 5-Methyl-2-phenyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 25 2-Methyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 26 2,5-Dimethyl-1-[2-(2-thienyl)-thiazol-4-ylmethyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 27 2,5-Dimethyl-1-[2-(3-chlorophenyl)-thiazol-4-ylmethyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 28 2,5-Dimethyl-1-[2-(4-chlorophenyl)-thiazol-4-ylmethyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 29 1-[2-(3-Fluoro-phenyl)-thiazol-4-ylmethyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 30 2,5-Dimethyl-1-(2-m-tolyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 31 2,5-Dimethyl-1-(2-pyridin-3-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 32 2,5-Dimethyl-1-(2-pyridin-4-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 33 2,5-Dimethyl-1-(3-methoxyphenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 34 2,5-Dimethyl-1-(4-methoxyphenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 35 2,5-Dimethyl-1-(2-p-tolyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 36 2,5-Dimethyl-1-(2-pyridin-2-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 37 2,5-Dimethyl-1-(2-thiophen-3-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 38 1-(2-Benzyl-thiazol-4-ylmethyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 39 2,5-Dimethyl-1-(2-furan-3-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 40 2,5-Dimethyl-1-(2-pyrazin-2-yl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 41 1-[2-(4-Ethoxy-phenyl)-thiazol-4-ylmethyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 42 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid [(R)-1-(4-aminomethyl-phenyl)-ethyl]-amide


name: US9670157, 43 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid (6-aminomethyl-pyridin-3-ylmethyl)-amide


name: US9670157, 44 1-[2-(3-Fluoro-phenyl)-thiazol-4-ylmethyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid (6-aminomethyl-pyridin-3-ylmethyl)-amide


name: US9670157, 45 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-3-fluoro-benzylamide


name: US9670157, 46 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-3-methyl-benzylamide


name: US9670157, 47 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-fluoro-benzylamide


name: US9670157, 48 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-((R)-1-amino-ethyl)-benzylamide


name: US9670157, 49 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-chloro-benzylamide


name: US9670157, 50 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-trifluoromethyl-benzylamide


name: US9670157, 52 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid [1-(4-aminomethyl-phenyl)-cyclopropyl]-amide


name: US9670157, 53 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-3-methoxy-benzylamide


name: US9670157, 54 2,5-Dimethyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-methoxy-benzylamide


name: US9670157, 55 1-Benzyl-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 56 1-Benzyl-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-chloro-benzylamide


name: US9670157, 57 1-Benzyl-5-methyl-2-phenyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 58 1-(3-Ethoxy-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 59 1-(4-Ethoxy-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 60 1-(4-Benzyloxy-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 61 1-(4-Methoxy-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 62 1-(3-Carbamoyl-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 63 1-(4-Carbamoyl-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 64 1-(3-Cyano-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 65 1-(4-Cyano-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 66 1-(3-Aminomethyl-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 67 1-(4-Aminomethyl-benzyl)-2,5-dimethyl-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 68 1-[4-(Acetylamino-methyl)-benzyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 69 1-Biphenyl-3-ylmethyl-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 70 1-Biphenyl-4-ylmethyl-2,5-dimethyl-1H-pyrrole-3-carboxylic acid4-aminomethyl-benzylamide


name: US9670157, 71 2,5-Dimethyl-1-(3-pyridin-3-yl-benzyl)-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 72 2,5-Dimethyl-1-(3-pyridin-4-yl-benzyl)-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 73 2,5-Dimethyl-1-(3-morpholin-4-yl-benzyl)-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 74 2,5-Dimethyl-1-(3-piperidin-1-yl-benzyl)-1H-pyrrole-3-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 75 5-Benzyl-1,4-dimethyl-1H-pyrrole-2-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 77 5-Benzyl-1-ethyl-4-methyl-1H-pyrrole-2-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 78 5-Benzyl-4-methyl-1-propyl-1H-pyrrole-2-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 79 1-(4-Isopropylcarbamoyl-benzyl)-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 80 5-Methyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrazole-4-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 81 3-Methyl-1-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrazole-4-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 82 1-(2-Phenyl-thiazol-4-ylmethyl)-5-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 83 1-(2-Phenyl-thiazol-4-ylmethyl)-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 84 1-Benzyl-3-phenyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 85 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 86 1-[4-(3,5-Dimethyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 87 1-[4-(Piperidine-1-carbonyl)-benzyl]-1H-pyrazole-4-carboxylicacid 4-aminomethyl-benzylamide


name: US9670157, 88 1-(4-Phenoxy-benzyl)-1H-[1,2,4]triazole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 89 1-[4-(2-Oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 90 2,5-Dimethyl-1-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 91 2,5-Dimethyl-1-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 92 1-Ethyl-4-methyl-5-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 93 1-Ethyl-4-methyl-5-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 94 2,5-Dimethyl-1-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 95 1-Ethyl-4-methyl-5-[4-(2-oxo-2H-pyridin-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 96 2,5-Dimethyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 97 2,5-Dimethyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 98 2,5-Dimethyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 99 1-Ethyl-4-methyl-5-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 100 1-Ethyl-4-methyl-5-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 101 2,5-Dimethyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 102 1-Ethyl-4-methyl-5-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 103 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 104 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-imidazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 105 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-imidazole-4-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 107 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-imidazole-4-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 108 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-[1,2,3]triazole-4-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 109 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-[1,2,3]triazole-4-carboxylic acid 4-aminomethyl-2-methyl-benzylamide


name: US9670157, 110 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-[1,2,3]triazole-4-carboxylic acid 4-(1-amino-cyclopropyl)-benzylamide


name: US9670157, 111 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 112 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-imidazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 113 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-1H-[1,2,3]triazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 114 3-Methyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 116 3,5-Dimethyl-1-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 117 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-3-fluoro-benzylamide


name: US9670157, 118 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 119 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-benzyl]-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-3-fluoro-2-methyl-benzylamide


name: US9670157, 121 1-Ethyl-4-methyl-5-[4-(4-methyl-pyrazol-1-ylmethyl)-benzyl]-1H-pyrrole-2-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 123 1-Ethyl-4-methyl-5-(2-phenyl-thiazol-4-ylmethyl)-1H-pyrrole-2-carboxylic acid 4-aminomethyl-benzylamide


name: US9670157, 124 3-Methyl-1-(2-methyl-quinolin-6-ylmethyl)-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 125 5-Methyl-1-(2-methyl-quinolin-6-ylmethyl)-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 126 1-(2-Methyl-quinolin-6-ylmethyl)-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 127 1-(2-Methyl-quinolin-6-ylmethyl)-5-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 128 2,5-Dimethyl-1-(2-methyl-quinolin-6-ylmethyl)-1H-pyrrole-3-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: US9670157, 129 1-(2-Pyrrolidin-1-yl-pyridin-4-ylmethyl)-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid 4-aminomethyl-2,6-dimethyl-benzylamide


name: 4-(3-Carbamoyl-5-pyridin-4-yl-1h-pyrrol-2-yl)-piperidine-1-carboxylic acid tert-butyl ester


name: US9670193, 4 N-benzyl-5-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)pyrimidin-2-amine (TFA-salt)


name: US9670193, 43 N-(Pyridin-4-ylmethyl)-2-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)pyrimidin-5-amine (TFA salt)


name: US9670196, 1.1 (1S,4R or 1R,4S)-methyl 4-(5-(3-((6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)amino)-5-methylphenyl)thiazol-2-yl)-4-hydroxy-2,2-dimethylcyclohexanecarboxylate


name: US9670196, 1.2 (1S,4R or 1R,4S)-4-(5-(3-((6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)amino)-5-methylphenyl)thiazol-2-yl)-4-hydroxy-2,2-dimethylcyclohexanecarboxylic acid


name: US9670196, 1.4 (R or S)-5-hydroxy-5-(5-(6-((2-methoxy-1,7-naphthyridin-6-yl)amino)-4-methylpyridin-2-yl)thiazol-2-yl)-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid


name: US9670196, 1.5 4-(1-(5-(6-(furo[3,2-b]pyridin-5-ylamino)-4-methylpyridin-2-yl)thiazol-2-yl)-1-hydroxyethyl)benzoic acid


name: US9670196, 1.7 (1S,4R or 1R,4S)-4-hydroxy-2,2-dimethyl-4-(5-(3-methyl-5-((4-methylfuro[3,2-d]pyrimidin-2-yl)amino)phenyl)thiazol-2-yl)cyclohexanecarboxylic acid


name: US9670196, 2.1 4-((5-(3-([1,2,4]triazolo[1,5-a]pyridin-2-ylamino)-5-methylphenyl)thiazol-2-yl)methyl)benzoic acid


name: US9670196, 2.2 (1S,4R or 1R,4S)-4-hydroxy-2,2-dimethyl-4-(5-{3-methyl-5-[(6-methyl-1,7-naphthyridin-8-yl)amino]phenyl}-1,3-thiazol-2-yl)cyclohexanecarboxylic acid


name: US9670196, 2.3 (R or S)-5-hydroxy-5-{5-[3-methyl-5-([1,2,4]triazolo[1,5-a]pyridin-2-ylamino)phenyl]-1,3-thiazol-2-yl}-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid


name: US9670196, 2.5 (R or S)-4-(1-hydroxy-1-{5-[3-methyl-5-([1,2,4]triazolo[1,5-a]pyridin-2-ylamino)phenyl]-1,3-thiazol-2-yl}ethyl)benzoic acid


name: RORC2 inverse agonist 66 [PMID: 30130103]


name: US9670208, Example 150 N-(1-methyl-1H-pyrazol-5-yl)-4-(3-neopentyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)pyrimidin-2-amine


name: US9670208, Example 169 4-(3-isobutyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine


name: US9670208, Example 211 4-(3-(2-fluorobenzyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-isopropylpyrimidin-2-amine


name: US9670208, Example 279 N-(1-methyl-1H-pyrazol-5-yl)-4-(3-neopentyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)pyridin-2-amine


name: US9670208, Example 411 4-([1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine


name: US9670210, Example 1 4-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)methyl]benzoic acid


name: US9670210, Example 2 N-{[1-(4-Fluorobenzyl)azetidin-3-yl]methyl}-trans-2-phenylcyclopropanamine


name: US9670210, Example 3 4-({4-[(trans-2-Phenylcyclopropyl)amino]piperidin-1-yl}methyl)benzoic acid


name: US9670210, Example 4 3-({4-[(trans-2-Phenylcyclopropyl)amino]piperidin-1-yl}methyl)benzoic acid


name: US9670210, Example 5 1-(4-Fluorobenzyl)-N-(trans-2-phenylcyclopropyl)piperidin-4-amine


name: US9670210, Example 6 4-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)methyl]benzonitrile


name: US9670210, Example 7 3-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)methyl]benzonitrile


name: US9670210, Example 8 (1-(3-Fluorobenzoyl)-4-{[(trans-2-phenylcyclopropyl)amino]methyl}piperidin-4-yl)acetonitrile


name: US9670210, Example 9 (1-(3-Fluorobenzyl)-4-{[(trans-2-phenylcyclopropyl)amino]methyl}piperidin-4-yl)acetonitrile


name: US9670210, Example 12 1-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)carbonyl]piperidine-4-carbonitrile


name: US9670210, Example 14 N-({1-[(3-Phenoxypiperidin-1-yl)carbonyl]azetidin-3-yl}methyl)-trans-2-phenylcyclopropanamine


name: US9670210, Example 15 N-({1-[(3-Methoxypiperidin-1-yl)carbonyl]azetidin-3-yl}methyl)-trans-2-phenylcyclopropanamine


name: US9670210, Example 17 4-Phenyl-1-[(3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidin-1-yl)carbonyl]piperidin-4-ol


name: US9670210, Example 19 N-(2-Fluorophenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 20 N-(3-Fluorophenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 21 N-(4-Fluorophenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 22 N-(4-Methoxyphenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 23 N-(3-Methoxyphenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 24 N-(2-Methoxyphenyl)-3-{[(trans-2-phenylcyclopropyl)amino]methyl}azetidine-1-carboxamide


name: US9670210, Example 25 4-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)carbonyl]benzonitrile


name: US9670210, Example 26 3-[(3-{[(trans-2-Phenylcyclopropyl)amino]methyl}azetidin-1-yl)carbonyl]benzonitrile


name: US9670210, Example 27 N-{[1-(3-Methoxybenzoyl)azetidin-3-yl]methyl}-trans-2-phenylcyclopropanamine


name: US9670210, Example 28 N-{[1-(4-Fluorobenzoyl)azetidin-3-yl]methyl}-trans-2-phenylcyclopropanamine


name: US9670210, Example 29 N-{[1-(3-Fluorobenzoyl)azetidin-3-yl]methyl}-trans-2-phenylcyclopropanamine


name: US9670210, Example 30 Trans-2-phenyl-N-[(1-{[4-(trifluoromethoxy)phenyl]sulfonyl}azetidin-3-yl)methyl]cyclopropanamine


name: US9670210, Example 31 1-{[4-(4-fluorobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 32 1-{[4-(4-fluorobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 35 1-{[4-(methoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 36 1-{[4-(methoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 37 1-{[4-(methoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopentanecarboxylic acid


name: US9670210, Example 38 (1R,2S) inverted question markN-[(4-(methoxymethyl)-1-{[(2S)-1-methylpyrrolidin-2-yl]carbonyl}piperidin-4-yl)methyl]-2-phenylcyclopropanamine


name: US9670210, Example 39 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-imidazol-4-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 41 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methylpiperidin-4-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 42 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-pyrazol-3-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 43 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(4-methylpiperazin-1-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 44 1-{[4-methyl-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 45 1-{[4-methyl-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 46 (1R,2S) inverted question markN-({4-methyl-1-[(1-methyl-1H-pyrazol-3-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 47 (1R,2S) inverted question markN-({4-methyl-1-[(1-methyl-1H-imidazol-4-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 52 5-{[4-methyl-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}pyrimidin-2-amine


name: US9670210, Example 53 1-{[4-[4-(cyanomethyl)benzyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 54 1-{[4-[4-(cyanomethyl)benzyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 55 1-{[4-(4-cyanobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 56 1-{[4-(3-cyanobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 57 1-{[4-(3-cyanobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 58 trans-4-{[4-(3-cyanobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclohexanecarboxylic acid


name: US9670210, Example 59 3-{[1-(3-methoxybenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-4-yl]methyl}benzoic acid


name: US9670210, Example 62 4-{[4-(methoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}benzoic acid


name: US9670210, Example 63 1-{[4-({[(1R,2S)-2-(4-fluorophenyl)cyclopropyl]amino}methyl)-4-(methoxymethyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 64 1-{[4-({[(1R,2S)-2-(2-fluorophenyl)cyclopropyl]amino}methyl)-4-(methoxymethyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 65 1-{[4-({[(1R,2S)-2-(3,4-difluorophenyl)cyclopropyl]amino}methyl)-4-(methoxymethyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 66 1-{[4-(methoxymethyl)-4-({[2-(2-methoxyphenyl)cyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 67 1-{[4-(methoxymethyl)-4-({[2-(4-methoxyphenyl)cyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 68 1-{[4-(methoxymethyl)-4-(1-{[(1R,2S)-2-phenylcyclopropyl]amino}ethyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 69 1-{[4-[(6-methoxypyridin-3-yl)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 70 1-{[4-(ethoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 71 1-{[4-(ethoxymethyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 72 1-{[4-[(benzyloxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 73 1-{[4-[(benzyloxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 74 1-{[4-(4-cyano-2-fluorobenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 75 1-{[4-[(2-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 76 1-{[4-[(2-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 77 1-{[4-[(3-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 78 1-{[4-[(3-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 79 1-{[4-[(2-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 80 1-{[4-[(3-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 81 1-{[4-[(4-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 82 1-{[4-[(4-cyano-2-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 83 1-{[4-[(2-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 84 1-{[4-[(3-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 85 1-{[4-[(4-cyanophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 86 1-{[4-[(4-cyano-2-fluorophenoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 87 1-{[4-{[(5-fluoropyridin-2-yl)oxy]methyl}-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 89 1-{[4-{[(3-fluoropyridin-2-yl)oxy]methyl}-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 92 1-{[4-[(cyclobutylmethoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 93 1-{[4-[(cyclobutylmethoxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 94 1-{[4-[(cyclohexyloxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 95 1-{[4-[(cyclohexyloxy)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 96 1-{[4-[(5-fluoropyridin-2-yl)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 97 1-{[4-[(5-fluoropyridin-2-yl)methyl]-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 98 1-{[4-(4-methoxybenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclopropanecarboxylic acid


name: US9670210, Example 99 1-{[4-(4-methoxybenzyl)-4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)piperidin-1-yl]methyl}cyclobutanecarboxylic acid


name: US9670210, Example 104 (1R,2S) inverted question markN-{[1-{[1-(2-methoxyethyl)-1H-pyrazol-4-yl]carbonyl}-4-(methoxymethyl)piperidin-4-yl]methyl}-2-phenylcyclopropanamine


name: US9670210, Example 105 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-pyrazol-4-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 113 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(4-methoxypiperidin-1-yl)carbonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 114 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 115 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-pyrazol-5-yl)sulfonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


name: US9670210, Example 116 (1R,2S) inverted question markN-({4-(methoxymethyl)-1-[(1-methyl-1H-pyrazol-3-yl)sulfonyl]piperidin-4-yl}methyl)-2-phenylcyclopropanamine


A pyrimidine compound having a 2-methoxy-4-(4-methylpiperazin-1-yl)anilino group at the 2-position, a 3-(acryloylamino)phenoxy group at the 4-position, and a chloro substituent at the 5-position.


name: A9UEZ6_HUMAN non-specific protein-tyrosine kinase (trembl)


TLR2_HUMAN Toll-like receptor 2 (sprot)

A Toll-like receptor 2 that is encoded in the genome of human.


name: KCNN4_HUMAN Intermediate conductance calcium-activated potassium channel protein 4 (sprot)

description: An intermediate conductance calcium-activated potassium channel protein 4 that is encoded in the genome of human.


name: Acetic acid 4-[4-chloro-3-(4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-1-yl)-phenoxy]-butyl ester


name: Process for preparing 1-(2-fluorophenyl)-5-{2-[2-(2-methoxyethoxyl)phenyl]phenyl}-1h-1,2,3,4-tetrazole


name: Process for preparing 5-{2-[2-(fluoromethoxy)phenyl]phenyl}-1-(2-fluorophenyl)-1h-1,2,3,4-tetrazole


name: Process for preparing 2-{2-[1-(2-fluorophenyl)-1h-1,2,3,4-tetrazol-5-yl]phenyl}benzaldehyde


name: Process for preparing 2-{2-[1-(2-fluorophenyl)-1h-1,2,3,4-tetrazol-5-yl]phenyl}-n,n-dimethylaniline


name: Process for preparing (2-{2-[1-(2-fluorophenyl)-1h-1,2,3,4-tetrazol-5-yl]phenyl}phenyl)methanol


name: Process for preparing 5-{2-[2-(difluoromethyl)phenyl]phenyl}-1-(2-fluorophenyl)-1h-1,2,3,4-tetrazole


name: Process for preparing 2-{2-[1-(2-fluorophenyl)-1h-1,2,3,4-tetrazol-5-yl]phenyl}-n-(2-methoxyethyl)aniline


name: Process for preparing 1-(2-chlorophenyl)-5-[2-(2-fluorophenyl)phenyl]-1h-1,2,3,4-tetrazole


name: Process for preparing 1-(2-chlorophenyl)-5-[2-(2-methoxyphenyl)phenyl]-1h-1,2,3,4-tetrazole


name: Process for preparing 1-(2-methoxyphenyl)-5-[2-(2-methoxyphenyl)phenyl]-1h-1,2,3,4-tetrazole


name: Process for preparing 2-{5-[2-(2-methoxyphenyl)phenyl]-1h-1,2,3,4-tetrazol-1-yl}phenol


name: Process for preparing 5-[2-(2-fluorophenyl)phenyl]-1-(2-methoxyphenyl)-1h-1,2,3,4-tetrazole


name: Process for preparing 2-{5-[2-(2-methoxyphenyl)phenyl]-1h-1,2,3,4-tetrazol-1-yl}benzonitrile


name: Process for preparing 1-[2-(difluoromethoxy)phenyl]-5-[2-(2-fluorophenyl)phenyl]-1h-1,2,3,4-tetrazole


name: Process for preparing 1-[2-(difluoromethoxy)phenyl]-5-[2-(2-methoxyphenyl)phenyl]-1h-1,2,3,4-tetrazole


name: Process for preparing 2-(5-{2-[2-(difluoromethoxy)phenyl]phenyl}-1h-1,2,3,4-tetrazol-1-yl)benzonitrile


name: Process for preparing 1-phenyl-5-(2-phenylphenyl)-1h-1,2,3,4-tetrazole


name: AKA7G_HUMAN A-kinase anchor protein 7 isoform gamma (sprot)


name: 6-{[(1r)-1-Cyclobutylethyl] amino}-8-(1,3-oxazol-2-yl)-7-[4-(trifluoromethyl) benzyl]-7h-purine-2-carboxylic acid


name: 6-{[(1r)-1-Cyclobutylethyl] amino}-8-(1,3-thiazol-2-yl)-7-[4-(trifluoromethyl) benzyl]-7h-purine-2-carboxylic acid


name: Sodium 6-chloro-7-(4-(4-chloro-2-(2-methoxyethoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(4-chloro-2-(trifluoromethoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(2-(4-chlorophenoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(4-chloro-2-(4-chlorophenoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(2-(3-chlorophenoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(2-(2-chlorophenoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(4-chloro-2-(3-chlorophenoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(4-chloro-2-(2-fluoroethoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: Sodium 6-chloro-7-(4-(4-chloro-2-(3-fluoropropoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylate


name: 7-(4-((1-(4-Chlorophenyl) cyclopropyl)methylcarbamoyl) phenoxy)-6-cyanochroman-4-carboxylic acid


name: 6-Chloro-7-(4-(4-(difluoromethoxy) phenethylcarbamoyl)phenoxy) chroman-4-carboxylic acid


name: 6-chloro-7-(4-((5-chloro-2,3-dihydro-1H-inden-1-yl) methylcarbamoyl)phenoxy) chroman-4-carboxylic acid


name: 6-Chloro-7-(4-(2-cyclopropyl-4-(trifluoromethyl) phenethylcarbamoyl)phenoxy) chroman-4-carboxylic acid


name: Preparation of 3-Fluoro-4-[4-fluoro-1-(2,5-difluorobenzyl)-1H-indazol-3-yl]benzoic acid (3A)


name: Preparation of 5-fluoro-4-(4-fluoro-1-(2-methyl-6-(trifluoromethyl)benzyl)-1H-indazol-3-yl)-2-hydroxybenzoic acid (8A) and 5-fluoro-4-(4-fluoro-1-(2-(trifluoromethyl)benzyl)-1H-indazol-3-yl)-2-hydroxybenzoic acid (8B)


name: Preparation of sodium 4-(1-(2-chloro-6-(trifluoromethyl)benzyl)-4-fluoro-6-(3-methoxyazetidine-1-carbonyl)-1H-indazol-3-yl)-5-fluoro-2-hydroxybenzoate (10A)


name: NMDE2_HUMAN Glutamate receptor ionotropic, NMDA 2B (sprot)

description: A glutamate receptor ionotropic, NMDA 2B that is encoded in the genome of human.


name: Methyl 4-[({5-hydroxy-5-phenyl-octahydrocyclopenta[c] pyrrol-2-yl}carbonyl)amino] benzoate


name: 6-Methoxy-5-[(S)-3 ((S)-2-methylamino-propionylamino)-2-oxo-5-(5-oxo-hexanoyl)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-ylmethyl]-naphthalene-2-carboxylic acid methyl ester hydrochloride


name: Preparation of 2-(7-(5-chloro-4-(2-(isopropylsulfonyl)phenylamino)pyrimidin-2 yl)amino)-6-methoxy-3,4-dihydroisoquinolin-2(1H)-yl)-N, N-dimethylacetamide


name: Preparation of 5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(7-isopropoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin 6 yl)pyrimidine-2,4-diamine


name: HBSAG_HBVD3 Large envelope protein (sprot)


P2RX7_MOUSE P2X purinoceptor 7 (sprot)

A P2X purinoceptor 7 that is encoded in the genome of mouse.


IL17_HUMAN Interleukin-17A (sprot)

An interleukin-17A that is encoded in the genome of human.


IL17F_HUMAN Interleukin-17F (sprot)

An interleukin-17F that is encoded in the genome of human.


IL21_HUMAN Interleukin-21 (sprot)

An interleukin-21 that is encoded in the genome of human.


IL22_HUMAN Interleukin-22 (sprot)

An interleukin-22 that is encoded in the genome of human.


name: Preparation of racemic 4-{[6-chloro-4''-(3-chloro-2-fluoro-phenyl)-2''-(1-fluoromethyl-cyclopropylmethyl)-2-oxo-1,2-dihydro-spiro[indole-3,3''-pyrrolidin]e-5''-carbonyl]-amino}-3-methoxy-benzoic acid methyl ester


name: Preparation of racemic 4-{[6-chloro-4''-(3-chloro-2-fluoro-phenyl)-2''-(1-fluoromethyl-cyclopropyl methyl)-2-oxo-1,2-dihydro-spiro[indole-3,3''-pyrrolidin]e-5''-carbonyl]-amino}-3-methoxy-benzoic acid


name: Preparation of racemic 6-chloro-4''-(3-chloro-2-fluoro-phenyl)-2''-(1-fluoromethyl-cyclopropyl methyl)-2-oxo-1,2-dihydro-spiro[indole-3,3''-pyrrolidine]-5-carboxylic acid (4-carbamoyl-2-methoxy-phenyl)-amide


name: 2-(2-Amino-ethylamino)-thieno[3,2-d]pyrimidine-7-carboxylic acid (1-methyl-1H-benzoimidazol-4-yl)-amide trifluoroacetate


name: 2-(Azetidin-3-ylamino)-thieno[3,2-d]pyrimidine-7-carboxylic acid (1-methyl-1H-benzoimidazol-4-yl)-amide hydrochloride


name: I22R2_HUMAN Interleukin-22 receptor subunit alpha-2 (sprot)

description: An interleukin-22 receptor subunit alpha-2 that is encoded in the genome of human.


name: FFAR4_HUMAN Free fatty acid receptor 4 (sprot)

description: A free fatty acid receptor 4 that is encoded in the genome of human.


name: ACMSD_HUMAN 2-amino-3-carboxymuconate-6-semialdehyde decarboxylase (sprot)

description: A 2-amino-3-carboxymuconate-6-semialdehyde decarboxylase that is encoded in the genome of human.


name: AGTR2_HUMAN Type-2 angiotensin II receptor (sprot)

description: An angiotensin II receptor 2 that is encoded in the genome of human.


name: (R)-5-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-4''-methoxy-1 inverted question mark,2 inverted question mark,3 inverted question mark,6 inverted question mark-tetrahydro-[3,3'':6'',4 inverted question mark-terpyridin]-6-amine


name: 5-((R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5''-methoxy-3 inverted question mark-methyl-1 inverted question mark,2 inverted question mark,3 inverted question mark,6 inverted question mark-tetrahydro-[3,3'':6'',4 inverted question mark-terpyridin]-6-amine


name: BLAB_SERMA Metallo-beta-lactamase type 2 (sprot)


name: BLAN1_KLEPN Metallo-beta-lactamase type 2 (sprot)

description: A protein that is a translation product of any of the plasmid-encoded copies of the blaNDM-1 gene in Klebsiella pneumoniae.


name: 3-(6-Aminopyridin-3-yl)-2-(1H-tetrazol-5-yl)benzene sulfonamide, TFA salt


name: (S)-2-amino-4-methyl-N inverted question mark((R)-5-methyl-5H-chromeno[3,4-c]pyridin-8-yl)pentanamide


name: (S)-2-amino-4-methyl-N inverted question mark((S)-5-methyl-5H-chromeno[3,4-c]pyridin-8-yl)pentanamide


name: CD36_RAT Platelet glycoprotein 4 (sprot)

description: A protein that is a translation product of the Cd36 gene in rat.


name: Synthesis of (S)-5-cyclopropyl-4-((1-(1-(3,5-dichlorophenyl)ethyl)-4-fluoropiperidin-4-yl)methoxy)-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-(((1R,3r,5S)-3-(3-chloro-2-fluoro-5-(trifluoromethyl)phenoxy)-8-azabicyclo[3.2.1]octan-8-yl)methyl)-5-cyclopropyl-N-(cyclopropylsulfonyl)-2-fluorobenzamide, trifluoroacetic acid salt


name: Synthesis of 4-(((1R,3r,5S)-3-(3-chloro-5-(trifluoromethoxy)phenoxy)-8-azabicyclo[3.2.1]octan-8-yl)methyl)-5-cyclopropyl-N-(cyclopropylsulfonyl)-2-fluorobenzamide, trifluoroacetic acid salt


name: Synthesis of 5-cyclopropyl-2-fluoro-N-(methylsulfonyl)-4-((4-(3-(trifluoromethyl)phenoxy)piperidin-1-yl)methyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-(4-chlorophenoxy)pyridin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-(2-chloro-4-fluorophenoxy)pyridin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide trifluoroacetic acid salt


name: Synthesis of 4-((4-(2-chloro-4-fluorophenoxy)pyridin-1-yl)methyl)-5-cyclopropyl-N-(cyclopropylsulfonyl)-2-fluorobenzamide, trifluoroacetic acid salt


name: Synthesis of 5-cyclopropyl-4-((4-(3,4-dichlorophenoxy)piperidin-1-yl)methyl)-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt)


name: Synthesis of 5-cyclopropyl-4-((4-((3,5-dichlorobenzyl)oxy)piperidin-1-yl)methyl)-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 5-cyclopropyl-2-fluoro-4-((4-(fluoromethyl)-4-(4-fluorophenyl)piperidin-1-yl)methyl)-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 5-cyclopropyl-2-fluoro-4-((4-(4-fluorophenyl)-4-(methoxymethyl)piperidin-1-yl)methyl)-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 5-cyclopropyl-4-((4-(3,5-dichlorobenzyl)piperazin-1-yl)methyl)-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-(4-chloro-3-(trifluoromethyl)phenoxy)piperidin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-((5-chloro-4-(trifluoromethyl)pyridin-2-yl)oxy)piperidin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-((3-chloro-5-(trifluoromethyl)pyridin-2-yl)oxy)piperidin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: Synthesis of 4-((4-(3-Chloro-2-fluoro-5-(trifluoromethyl)phenoxy)piperidin-1-yl)methyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide, trifluoroacetic acid salt


name: GP139_HUMAN Probable G-protein coupled receptor 139 (sprot)

description: A probable G-protein coupled receptor 139 that is encoded in the genome of human.


name: 2-{5-Amino-1-[4-(3-cyano-phenoxy)-2-methyl-phenyl]-1h-pyrazole-4-carbonyl}-1h-indole-5-carboxylic acid methyl ester


name: 2-{5-Amino-1-[2-chloro-4-(2-dimethylcarbamoyl-phenoxy)-phenyl]-1h-pyrazole-carbonyl}-1h-indole-5-carboxylic acid (1-methyl-pyrrolidin-3-y1)-amide acetic acid salt


name: 2-{5-Amino-1-[2-chloro-4-(2-dimethylcarbamoyl-phenoxy)-phenyl]-1h-pyrazole-4-carbonyl}-1h-indole-5-carboxylic acid (2-methylamino-ethyl)-amideacetic acid salt


WNT3A_HUMAN Protein Wnt-3a (sprot)

A protein Wnt-3a that is encoded in the genome of human.


name: NDUV1_BOVIN NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial (sprot)

description: An NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial that is encoded in the genome of cow.


name: US9714221, Example 219N/A*: Not available. Prodrug of example 75


name: HOGA1_HUMAN 4-hydroxy-2-oxoglutarate aldolase, mitochondrial (sprot)

description: A 4-hydroxy-2-oxoglutarate aldolase, mitochondrial that is encoded in the genome of human.


name: Synthesis of N-(7-(2-(adamantan-2-yl)ethoxy)-6-cyclopropyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methanesulfonamide 7)


name: AKCL2_HUMAN 1,5-anhydro-D-fructose reductase (sprot)

description: A 1,5-anhydro-D-fructose reductase that is encoded in the genome of human.


name: (E)-3-(4-((2-(4-chlorophenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(3-fluorophenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((6-hydroxy-2-(2-(trifluoromethyl)-phenyl)benzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2-chlorophenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(4-fluoro-2-methylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2,3-dimethylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2,5-dimethylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((6-hydroxy-2-(3-hydroxy-2-methyl-phenyl)benzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2-ethylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2-acetylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(2-(tert-butyl)phenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(4-(tert-butyl)phenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-3-(4-((2-(3,5-dimethylphenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylic acid


name: (E)-methyl 3-(4-((2-(4-fluorophenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy) phenyl)-acrylate


name: (E)-3-(4-((2-(3-fluoro-2-(trifluoromethyl) phenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy)phenyl)acrylic acid


name: (E)-3-(4-((2-(5-fluoro-2-(trifluoromethyl) phenyl)-6-hydroxybenzo[b] thiophen-3-yl)oxy)phenyl)acrylic acid


name: (E)-3-(4-((6-hydroxy-2-(3-isopropylphenyl) benzo[b] thiophen-3-yl)oxy)phenyl)acrylic acid


name: (E)-2-(4-((6-hydroxy-2-(2-isopropylphenyl)benzo [b]thiophen-3-yl)oxy)benzylidene) butanoic acid


name: (E)-2-(4-((6-hydroxy-2-(4-hydroxyphenyl)benzo [b]thiophen-3-yl)oxy)benzylidene) butanoic acid


name: (E)-3-(4-((6-hydroxy-2-(2-isopropylphenyl)benzo [b]thiophen-3-yl)(methyl)amino)phenyl) acrylic acid


name: FFAR2_HUMAN Free fatty acid receptor 2 (sprot)

description: A free fatty acid receptor 2 that is encoded in the genome of human.


name: LCAP_RAT Leucyl-cystinyl aminopeptidase (sprot)

description: A leucyl-cystinyl aminopeptidase that is encoded in the genome of rat.


name: LCAP_HUMAN Leucyl-cystinyl aminopeptidase (sprot)

description: A leucyl-cystinyl aminopeptidase that is encoded in the genome of human.


name: Q72502_9HIV1 Envelope glycoprotein gp160 (trembl)


name: VIF_HV1N5 Virion infectivity factor (sprot)


name: ENV_HV1BR Envelope glycoprotein gp160 (sprot)


name: ERG_HUMAN Transcriptional regulator ERG (sprot)

description: A transcriptional regulator ERG that is encoded in the genome of human.


name: US95556117, Example 1,4-Chloro-1H-indole-5-carboxylicacid ((S)-1-cyclohexyl-2-hydroxy-ethyl)-amide


name: US95556117, Example 2,4-Chloro-1H-indole-5-carboxylicacid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 4,4-Chloro-1H-indole-5-carboxylicacid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 5,4-Chloro-1H-indole-5-carboxylicacid [(S)-1-(4,4-difluoro-cyclohexyl)-2-hydroxy-ethyl]-amide


name: US95556117, Example 6,4-Chloro-1-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 7,4-Chloro-1-methyl-1H-indole-5-carboxylic acid ((S)-1-cyclohexyl-2-hydroxy-ethyl)-amide


name: US95556117, Example 8,4-Chloro-3-formyl-1H-indole-5-carboxylic acid ((S)-1-cyclohexyl-2-hydroxy-ethyl)-amide


name: US95556117, Example 9,4-Chloro-3-formyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 10,rac-4-Chloro-1H-indole-5-carboxylic acid (1-cycloheptyl-2-hydroxy-ethyl)-amide


name: US95556117, Example 11,4-Chloro-1H-indole-5-carboxylicacid [1-(2-trifluoromethyl-pyrimidin-5-yl)-


name: US95556117, Example 12,4-Chloro-1H-indole-5-carboxylicacid [1-(6-chloro-pyridin-3-yl)-cyclohexylmethyl]-amide


name: US95556117, Example 13,4-Chloro-1H-indole-5-carboxylicacid [1-(6-trifluoromethyl-pyridin-3-yl)-cyclohexylmethyl]-amide


name: US95556117, Example 15,4-Chloro-1H-indole-5-carboxylicacid [1-(4-chloro-phenyl)-cyclohexylmethyl]-amide


name: US95556117, Example 16,4-Chloro-1H-indole-5-carboxylicacid [1-(4-trifluoromethyl-phenyl)-cyclohexylmethyl]-amide


name: US95556117, Example 17,4-Chloro-1H-indole-5-carboxylicacid (1-pyridin-3-yl-cyclohexylmethyl)-amide


name: US95556117, Example 18,4-Chloro-1H-indole-5-carboxylicacid (1-pyridin-3-yl-cyclopentylmethyl)-amide


name: US95556117, Example 19,4-Chloro-1H-indole-5-carboxylicacid (1-pyridin-3-yl-cycloheptylmethyl)-amide


name: US95556117, Example 20,4-Chloro-7-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 21,4-Chloro-2-oxo-2,3-dihydro-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 22,4-Chloro-2-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 23,4-Chloro-7-iodo-3-methylsulfanyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 24,4-Chloro-7-methyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 25,4-Chloro-7-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 26,4-Chloro-3-fluoro-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 27,4-Methoxy-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 28,3,4-Dichloro-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: 1-{[(4-chloro-1H-indole-5-carbonyl)-amino]-methyl}-cyclohexane carboxylic acid methyl ester


name: 4-Chloro-1H-indole-5-carboxylic acid (1-hydroxymethyl-cyclohexyl methyl)-amide


name: 7-Amino-4-chloro-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexyl methyl)-amide


name: US95556117, Example 33,4-Chloro-3-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 35,4-Chloro-1H-indole-5-carboxylicacid (1-methylcarbamoyl-cyclohexylmethyl)-amide


name: (1-{[(4-chloro-1H-indole-5-carbonyl)-amino]-methyl}-cyclohexyl)-carbamic acid tert-butyl ester


name: US95556117, Example 38,4,6-Dichloro-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 39,4-Chloro-1H-indole-5-carboxylicacid (1-amino-cyclohexylmethyl)-amidehydrochloride


name: US95556117, Example 40,4-Chloro-6-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 41,4-Chloro-1H-indole-5-carboxylicacid (1-hydroxy-cyclopentylmethyl)-amide


name: US95556117, Example 42,4-Chloro-1H-indole-5-carboxylicacid (1-hydroxy-cyclooctylmethyl)-amide


name: US95556117, Example 43,4-Chloro-1H-indole-5-carboxylicacid (1-methoxy-cyclohexylmethyl)-amide


name: US95556117, Example 44,4-Chloro-1H-indole-5-carboxylicacid ((S)-1-cyclohexyl-ethyl)-amide


name: US95556117, Example 45,4-Chloro-1H-indole-5-carboxylicacid ((R)-1-cyclohexyl-ethyl)-amide


name: US95556117, Example 48,4-Chloro-1H-indole-5-carboxylicacid (1-dimethylamino-cyclohexylmethyl)-amide


name: US95556117, Example 50,3-Bromo-4-chloro-7-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 51,(1-{[(4-Chloro-1H-indole-5-carbonyl)-amino]-methyl}-cyclohexylsulfamoyl)-acetic acidmethyl ester


name: US95556117, Example 52,4-Chloro-7-isobutyl-1H-indol-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 53,4-Chloro-7-(3-methoxy-propyl)-1H-indole-5-carboxylic acid (1-hydroxy-cycloheptylmethyl)-amide


name: US95556117, Example 54,4-Chloro-7-isobutyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 55,4-Chloro-7-(3-methoxy-propyl)-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 56,4-Chloro-1H-indole-5-carboxylicacid [1-(2-hydroxy-ethanesulfonylamino)-cyclohexylmethyl]-amide


name: US95556117, Example 57,4-Methyl-1H-indole-5-carboxylicacid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 58,4-Chloro-1H-indole-5-carboxylicacid [1-(2-methyl-pyrimidin-5-yl)-cyclohexylmethyl]-amide


name: US95556117, Example 59,4-Chloro-7-methoxy-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 61,4-Chloro-7-methyl-1H-indole-5-carboxylic acid [4,4-difluoro-1-(2-methyl-pyrimidin-5-yl)-cyclohexylmethyl]-amide


name: US95556117, Example 62,4-Chloro-7-methyl-1H-indole-5-carboxylic acid [1-(2-methyl-pyrimidin-5-yl)-cyclohexylmethyl]-amide


name: US95556117, Example 63,4,7-Dimethyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 64,4-Methyl-1H-indole-5-carboxylicacid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 65,4-Ethyl-1H-indole-5-carboxylicacid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 69,7-Methyl-4-trifluoromethyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 70,7-Methyl-4-trifluoromethyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 71,4,7-Dimethyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 72,4-Chloro-7-ethyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 73,4-Chloro-7-ethyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 74,7-Chloro-4-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 75,7-Chloro-4-methyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 76,4-Chloro-7-methoxy-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 77,7-Methoxy-4-methyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 78,7-Methoxy-4-methyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 79,4-Chloro-7-ethoxy-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 80,4-Chloro-7-hydroxy-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 81,4-Chloro-7-ethoxy-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 82,4-Chloro-7-propyl-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 83,4-Chloro-7-propyl-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 87,4-Chloro-7-(2-hydroxy-ethoxy)-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 88,7-Acetyl-4-chloro-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 90,4,7-Difluoro-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 91,4,7-Difluoro-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 92,4-Fluoro-7-methoxy-1H-indole-5-carboxylic acid (1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 93,4-Fluoro-7-methoxy-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 94,4-Chloro-7-(2-ethoxy-ethyl)-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-amide


name: US95556117, Example 95,4-Chloro-7-(1-methoxy-1-methyl-ethyl)-1H-indole-5-carboxylic acid (4,4-difluoro-1-hydroxy-cyclohexylmethyl)-


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-4-(1H-pyrazol-3-yl) benzamide


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-6-(trifluoromethyl) nicotinamide


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-2-(4-methoxyphenyl) thiazole-4-carboxamide, 3 HCl


name: 2-(dimethylamino)-N-(6-(2-(4-fluorophenyl)imidazo[1,2-a] pyridin-3-yl)imidazo[1,2-b] pyridazin-2-yl) isonicotinamide


name: 2-amino-N-(6-(2-(4-fluorophenyl)imidazo[1,2-a] pyridin-3-yl)imidazo[1,2-b] pyridazin-2-yl) isonicotinamide


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-2-(trifluoromethyl) isonicotinamide


name: 3-fluoro-N-(6-(2-(4-fluorophenyl)imidazo[1,2-a] pyridin-3-yl)imidazo[1,2-b] pyridazin-2-yl) isonicotinamide


name: 5-chloro-N-(6-(2-(4-fluorophenyl)imidazo[1,2-a] pyridin-3-yl)imidazo[1,2-b] pyridazin-2-yl) nicotinamide


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-5-(thiophen-2-yl) nicotinamide


name: N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-yl) imidazo[1,2-b]pyridazin-2-yl)-2-(1H-imidazol-1-yl) acetamide


name: APC_HUMAN Adenomatous polyposis coli protein (sprot)

description: An adenomatous polyposis coli protein that is encoded in the genome of human.


name: PRI724; PRI 724; ICG001 isomer; ICG-001 isomer; ICG 001 isomer


name: CNBP1_HUMAN Beta-catenin-interacting protein 1 (sprot)

description: A beta-catenin-interacting protein 1 that is encoded in the genome of human.


ADEFOVIR

A member of the class of phosphonic acids that is methylphosphonic acid in which one of the methyl hydrogens has been replaced by a 2-(6-amino-9H-purin-9-yl)ethoxy group. An inhibitor of HIV-1 reverse transcriptase, the bis(t-butoxycarbonyloxymethyl) ester (dipivoxil ester) prodrug is used to treat chronic hepatitis B viral infection.


name: CSF1R_RAT Macrophage colony-stimulating factor 1 receptor (sprot)

description: A macrophage colony-stimulating factor 1 receptor that is encoded in the genome of rat.


name: INGR1_HUMAN Interferon gamma receptor 1 (sprot)

description: An interferon gamma receptor alpha chain that is encoded in the genome of human.


ITA8_HUMAN Integrin alpha-8 (sprot)

An integrin alpha-8 that is encoded in the genome of human.


ITB3_HUMAN Integrin beta-3 (sprot)

An integrin beta-3 that is encoded in the genome of human.


ITB5_HUMAN Integrin beta-5 (sprot)

An integrin beta-5 that is encoded in the genome of human.


ITB6_HUMAN Integrin beta-6 (sprot)

An integrin beta-6 that is encoded in the genome of human.


ITB8_HUMAN Integrin beta-8 (sprot)

An integrin beta-8 that is encoded in the genome of human.


name: TEP1_HUMAN Telomerase protein component 1 (sprot)

description: A telomerase protein component 1 that is encoded in the genome of human.


name: Synthesis of (S)-4-(2-(5-chloro-2-fluorophenyl)-5-ethylpyridin-4-ylamino)-N-(2-hydroxy propyl)nicotinamide


name: Synthesis of 4-[[2-(5-chloro-2-fluoro-phenyl)-5-isopropenyl-4-pyridyl]amino]-N-(2-hydroxy ethyl)pyridine-3-carboxamide


name: Synthesis of N-[(2S)-2-hydroxypropyl]-4-{[2-phenyl-5-(propan-2-yl)pyridin-4-yl]amino} pyridine-3-carboxamide


name: BMR1B_MOUSE Bone morphogenetic protein receptor type-1B (sprot)

description: A BMP receptor type-1B that is encoded in the genome of mouse.


name: ABHD2_MOUSE Monoacylglycerol lipase ABHD2 (sprot)

description: A monoacylglycerol lipase ABHD2 that is encoded in the genome of mouse.


name: ATA_ACIBT Adhesin Ata autotransporter (sprot)


name: GP160_HUMAN Probable G-protein coupled receptor 160 (sprot)

description: A probable G-protein coupled receptor 160 that is encoded in the genome of human.


name: SMYD2_HUMAN N-lysine methyltransferase SMYD2 (sprot)

description: An N-lysine methyltransferase SMYD2 that is encoded in the genome of human.


name: GRK5_HUMAN G protein-coupled receptor kinase 5 (sprot)

description: A G protein-coupled receptor kinase 5 that is encoded in the genome of human.


name: GRK1_HUMAN Rhodopsin kinase GRK1 (sprot)

description: A rhodopsin kinase GRK1 that is encoded in the genome of human.


name: GLYM_HUMAN Serine hydroxymethyltransferase, mitochondrial (sprot)

description: A serine hydroxymethyltransferase, mitochondrial that is encoded in the genome of human.


name: GLYC_HUMAN Serine hydroxymethyltransferase, cytosolic (sprot)

description: A serine hydroxymethyltransferase, cytosolic that is encoded in the genome of human.


name: PP2BC_HUMAN Serine/threonine-protein phosphatase 2B catalytic subunit gamma isoform (sprot)

description: A serine/threonine-protein phosphatase 2B catalytic subunit gamma isoform that is encoded in the genome of human.


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-methyl-1H-imidazol-2-yl)-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-(N-morpholino-ethyl)-1H-imidazol-2-yl)-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-(N-pyrrolidinyl-ethyl)-1H-imidazol-2-yl) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-5-(1-(N,N-Dimethyl-ethyl)-1H-imidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-5-(1-(3-hydroxypropyl)-1H-imidazol-2-yl)-4-methyl-2-(methylamino) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino) 5-(1-(pyridin-3-yl-ethyl)-1H-imidazol-2-yl) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-[3-(3,3,3-trifluoro-propyl)-3H-imidazol-2-yl]-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-1-(1H-Benzimidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino)pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-1-(1H-Benzimidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino) pentanoic acid]1 cyclosporin A


name: [(2S,3R,4S)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-3-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(2-methyl-thiazol-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-7-(5-Fluoro-pyridin-2-yl)-3-hydroxy-4-methyl-2-(methylamino)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(5-methoxy-pyridin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(2-methyl-pyridin-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A


name: [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrazin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A